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2025-04-15 加入
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Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases
3小时前
已完结
Discovery of Aryl Benzoyl Hydrazide Derivatives as Novel Potent Broad-Spectrum Inhibitors of Influenza A Virus RNA-Dependent RNA Polymerase (RdRp)
3小时前
已完结
Discovery of Pyrazolopyridine Derivatives as HPK1 Inhibitors
3小时前
已完结
Discovery of N-(2-chloro-5-(3-(pyridin-4-yl)-1H-pyrazolo[3,4-b]pyridin-5-yl)pyridin-3-yl)-4-fluorobenzenesulfonamide (FD274) as a highly potent PI3K/mTOR dual inhibitor for the treatment of acute myeloid leukemia
3小时前
已完结
Introduction of a carboxylic acid group into pyrazolylpyridine derivatives increased selectivity for inhibition of the 20-HETE synthase CYP4A11/4F2
3小时前
已完结
Structure-activity relationship study of 1,6-naphthyridinone derivatives as selective type II AXL inhibitors with potent antitumor efficacy
3小时前
已完结
Discovery of Potent, Orally Bioavailable, Tricyclic NLRP3 Inhibitors
4小时前
已完结
Discovery of Hepatitis B Virus Surface Antigen Suppressor GS-8873
4小时前
待确认
Discovery of Hepatitis B Virus Surface Antigen Suppressor GS-8873
4小时前
已完结
Structure-based design and synthesis of BML284 derivatives: A novel class of colchicine-site noncovalent tubulin degradation agents
4小时前
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