咪唑
蛋白酶
组合化学
化学
严重急性呼吸综合征冠状病毒2型(SARS-CoV-2)
病毒学
立体化学
药理学
2019年冠状病毒病(COVID-19)
生物化学
生物
医学
酶
内科学
疾病
传染病(医学专业)
作者
P. Huynh,Phatcharin Khamplong,Minh-Hoang Phan,Thanh-Phuc Nguyen,Phuong Ngoc Lan Vu,Quang-Vinh Tang,Phumin Chamsodsai,Supaphorn Seetaha,Truong L. Tuong,Thien Y. Vu,Duc-Duy Vo,Kiattawee Choowongkomon,Cam‐Van T. Vo
摘要
Novel asymmetric imidazole-4,5-dicarboxamide derivatives were synthesized, evaluated for SARS-CoV-2 M Pro inhibitory activity in vitro , and investigated for binding ability in silico .
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