Lv2
190 积分 2024-04-08 加入
Efficient Route for the Synthesis of Diverse Heteroannelated 5-Cyanopyridines
1个月前
已完结
Discovery of a first-in-class reversible DNMT1-selective inhibitor with improved tolerability and efficacy in acute myeloid leukemia
1个月前
已完结
DNMT1 binds HDAC2 and a new co-repressor, DMAP1, to form a complex at replication foci
1个月前
已完结
Novel ATR/PARP1 Dual Inhibitors Demonstrate Synergistic Antitumor Efficacy in Triple‐Negative Breast Cancer Models
2个月前
已完结
Discovery of Quinazoline-2,4(1H,3H)-dione Derivatives Containing 3-Substituted Piperizines as Potent PARP-1/2 Inhibitors─Design, Synthesis, In Vivo Antitumor Activity, and X-ray Crystal Structure Analysis
2个月前
已完结
Biocatalytic Synthesis and Structure Elucidation of Cyclized Metabolites of the Deacetylase Inhibitor Panobinostat (LBH589)
2个月前
已完结
Non-hydroxamate Histone Deacetylase Inhibitors
2个月前
已完结
Structure–Activity Relationship Studies of DNA Methyltransferase 1 Monovalent Degraders
4个月前
已完结
Recent Study of Dual HDAC/PARP Inhibitor for the Treatment of Tumor
4个月前
已完结
PARP inhibitors: A review of the pharmacology, pharmacokinetics, and pharmacogenetics
5个月前
已完结