Lv2
150 积分 2025-02-24 加入
Discovery of 1,2,3,4-Tetrahydrochromeno[3,4c]pyridin-5-one Derivatives as Novel MTHFD Inhibitors for the Treatment of Acute Myeloid Leukemia
28天前
已完结
Discovery of DN1679 as a Potent, Orally Bioavailable, and Highly Selective CDK12/13 Dual Degrader for the Treatment of Triple-Negative Breast Cancer
3个月前
已完结
Discovery of Benzodiazepinepyrimidine Scaffold Derivatives as Potent Doublecortin-Like Kinase 1 (DCLK1) Inhibitors for the Treatment of Acute Inflammatory Diseases
4个月前
已完结
Leveraging Dual-Ligase Recruitment to Enhance Protein Degradation via a Heterotrivalent Proteolysis Targeting Chimera
5个月前
已完结
Exploration of a Novel, Enamine-Solid-Base Catalyzed Aldol Condensation with C-Glycosidic Pyranoses and Furanoses
6个月前
已完结
Discovery of CYP1A1 Inhibitors for Host-Directed Therapy against Sepsis
7个月前
已完结
The V ilsmeier Reaction of Fully Conjugated Carbocycles and Heterocycles
9个月前
已完结
Visible-light-absorbing C–N cross-coupling for the synthesis of hydrazones involving C(sp2)–H/C(sp3)–H functionalization
9个月前
已完结