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10 积分 2025-09-04 加入
Synthesis of ( S )-3-amino-benzo[ b ][1,4]oxazepin-4-one via Mitsunobu and S N Ar reaction for a first-in-class RIP1 kinase inhibitor GSK2982772 in clinical trials
1小时前
已完结
A highly enantioselective acyl-Mannich reaction of isoquinolines with aldehydes promoted by proline derivatives: an approach to 13-alkyl-tetrahydroprotoberberine alkaloids
30天前
已完结
Predictable site-selective functionalization: Promoter group assisted para-halogenation of N-substituted (hetero)aromatics under metal-free condition
1个月前
已完结
Site-Selective C–H Functionalization of (Hetero)Arenes via Transient, Non-symmetric Iodanes
1个月前
已完结
Isoquinoline Kelch-like ECH-Associated Protein 1-Nuclear Factor (Erythroid-Derived 2)-like 2 (KEAP1-NRF2) Inhibitors with High Metabolic Stability
1个月前
已完结
Direct C4 Halogenation of Isoquinolines via a Boc2O-Mediated Dearomatization Strategy
1个月前
已完结
Total Syntheses of Cinchona Alkaloids via Photoredox-Catalyzed Deoxygenative Arylation
1个月前
已完结
Strategies and Synthetic Methods Directed Toward the Preparation of Libraries of Substituted Isoquinolines
1个月前
已完结
Preparation of 1,3‐disubstituted isoquinoline derivatives from N‐boc‐3‐substituted‐1,2‐dihydroisoquinolines
1个月前
已完结
32nd Symposium on Progress in Organic Reactions and Syntheses
1个月前
已关闭