Lv22
102 积分 2023-08-04 加入
Discovery of a brain-penetrant fourth-generation EGFR inhibitor to overcome the human triple (L858R/T790 M/C797S) mutation
1小时前
待确认
Top 20 Best-Selling Small-Molecule Neurology Drugs in 2024: Market, Indications, Pharmacology, Discovery, and Synthesis
3天前
已完结
Optimization of linear and cyclic peptide inhibitors of KEAP1-NRF2 protein-protein interaction
25天前
已完结
Identification of highly selective type II kinase inhibitors with chiral peptidomimetic tails
25天前
已完结
Switchable Nucleophilic Site Enables Expedient Synthesis of CF3-Containing Thiazoles and Allenes from 1,3-Enynes
25天前
已完结
Identification of Small Molecule Inhibitors and Ligand Directed Degraders of Calcium/Calmodulin Dependent Protein Kinase Kinase 1 and 2 (CaMKK1/2)
25天前
已完结
Discovery of Quinoxaline-Based P1–P3 Macrocyclic NS3/4A Protease Inhibitors with Potent Activity against Drug-Resistant Hepatitis C Virus Variants
25天前
已完结
Structure-based Discovery of Cell-Potent Peptidomimetic Inhibitors for Protein N-Terminal Methyltransferase 1
25天前
已完结
Microwave Assisted Synthesis and Antimicrobial Activity of Novel Pyrrolidine Derivatives
25天前
已完结
Discovery of (S)-N1-(thiazol-2-yl) pyrrolidine-1,2-dicarboxamide derivatives targeting PI3Ka/HDAC6 for the treatment of cancer
25天前
已完结