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62 积分 2024-01-27 加入
Cannabinoid receptor 1 ligands: Biased signaling mechanisms driving functionally selective drug discovery
15天前
已完结
Ensifentrine: First Approval
17天前
已完结
Conformationally Restricted Pleuromutilins via A Pyridinyl-Amide Tether Bias Peptidyl Transferase Center Engagement Enabling Broad-Spectrum Potency Against Multidrug-Resistant Bacteria
26天前
已关闭
The Use of Conformational Restriction in Medicinal Chemistry
1个月前
已完结
Allosteric Regulation and Inhibition of Coronavirus 3CLpro Revealed by HDX‐MS
2个月前
已完结
Methyl rosmarinate is an allosteric inhibitor of SARS-CoV-2 3 CL protease as a potential candidate against SARS-cov-2 infection
2个月前
已完结
Covalent-Allosteric Kinase Inhibitors
2个月前
已完结
Methyl rosmarinate is an allosteric inhibitor of SARS-CoV-2 3 CL protease as a potential candidate against SARS-cov-2 infection
2个月前
已完结
Cell‐Active, Irreversible Covalent Inhibitors Targeting a Surface‐Exposed Non‐Catalytic Lysine on Aurora a Kinase by Using Squarate Chemistry
2个月前
已完结
68Ga‐labeled Ciprofloxacin Conjugates as Radiotracers for Targeting Bacterial Infection
3个月前
已完结