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Lv11
20 积分
2024-08-13 加入
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Novel 1,3-Thiazole Analogues with Potent Activity against Breast Cancer: A Design, Synthesis, In Vitro, and In Silico Study
4小时前
已完结
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Design, Synthesis, and Biological Evaluation of 1-(Indolizin-3-yl)ethan-1-ones as CBP Bromodomain Inhibitors for the Treatment of Prostate Cancer
1个月前
已完结
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Structure-Based Discovery and Optimization of Furo[3,2c]pyridin-4(5H)one Derivatives as Potent and Second Bromodomain (BD2)-Selective Bromo and Extra Terminal Domain (BET) Inhibitors
1个月前
已完结
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Design, synthesis and biological evaluation of some new 2-Pyrazoline derivatives as potential anticancer agents
3个月前
已完结
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Identification of a 2‐phenylthiazole derivative acetylcholinesterase modulator with in vitro antitumor activity in breast cancer cells
3个月前
已完结
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Design, Synthesis, and Antitumor Activity Evaluation of 2-Phenylthiazole-5-Carboxylic Acid Derivatives Targeting Transactivation Response RNA-Binding Protein 2
3个月前
已完结
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Synthesis, characterization, anticancer, pharmacokinetics and molecular docking investigation of N (3)-alkyl incorporated-3-acetyl-4-hydroxycoumarin thiosemicarbazones and their copper(II) complexes
3个月前
已完结
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Synthesis, characterization, and anticancer potency of coumarin-derived thiosemicarbazones and their Copper(II) complexes
3个月前
已完结
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Discovery of a potent and selective CBP bromodomain inhibitor (Y08262) for treating acute myeloid leukemia
4个月前
已完结
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Fluorine in medicinal chemistry
4个月前
已完结