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1315 积分 2021-08-29 加入
Proteolysis targeting chimera (PROTAC) in drug discovery paradigm: Recent progress and future challenges
1小时前
待确认
Discovery of novel antagonists targeting the DNA binding domain of androgen receptor by integrated docking-based virtual screening and bioassays
1小时前
待确认
Discovery of LYA914, An Orally Bioavailable PROTAC Degrader Targeting the DNA Binding Domain of the Androgen Receptor for the Treatment of CRPC
2小时前
待确认
Modular PROTAC/IMiD Bifunctional Molecule Design for the Degradation of Synergistic Targets in the Treatment of Lymphoma
1天前
待确认
Time-resolved Förster Resonance Energy Transfer Assays for Measurement of Endogenous Phosphorylated STAT Proteins in Human Cells
7天前
已完结
Discovery of BRD9 Molecular Glue Degraders That Spare Cardiomyocytes
10天前
已完结
Template-assisted covalent modification underlies activity of covalent molecular glues
10天前
已完结
A Top-Down Design Approach for Generating a Peptide PROTAC Drug Targeting Androgen Receptor for Androgenetic Alopecia Therapy
29天前
已完结
Design and characterization of cereblon-mediated androgen receptor proteolysis-targeting chimeras
29天前
已完结
Proteolysis targeting chimera (PROTAC) in drug discovery paradigm: Recent progress and future challenges
29天前
已完结