Lv51
970 积分 2021-12-24 加入
Structure of mitochondrial pyruvate carrier and its inhibition mechanism
2小时前
已完结
“Angular” Spirocyclic Azetidines: Synthesis, Characterization, and Evaluation in Drug Discovery
1个月前
已完结
Discovery, Synthesis, and Biological Evaluation of Thiazoloquin(az)olin(on)es as Potent CD38 Inhibitors
2个月前
已完结
Discovery of 4-Amino-8-quinoline Carboxamides as Novel, Submicromolar Inhibitors of NAD-Hydrolyzing Enzyme CD38
2个月前
已完结
Small-molecule inhibition of Lats kinases may promote Yap-dependent proliferation in postmitotic mammalian tissues
3个月前
已完结
Development of an improved inhibitor of Lats kinases to promote regeneration of mammalian organs
3个月前
已完结
Small molecule LATS kinase inhibitors block the Hippo signaling pathway and promote cell growth under 3D culture conditions
3个月前
已完结
NIBR-LTSi is a selective LATS kinase inhibitor activating YAP signaling and expanding tissue stem cells in vitro and in vivo
3个月前
已完结
Discovery of Orally Efficacious Bridged Piperazines as smTNF Modulators
3个月前
已完结
Discovery of SD-436: A Potent, Highly Selective and Efficacious STAT3 PROTAC Degrader Capable of Achieving Complete and Long-Lasting Tumor Regression
3个月前
已完结