Lv4
468 积分 2021-04-15 加入
Discovery of a Potent (4R,5S)-4-Fluoro-5-methylproline Sulfonamide Transient Receptor Potential Ankyrin 1 Antagonist and Its Methylene Phosphate Prodrug Guided by Molecular Modeling
1天前
已完结
A Retrospective Look at the Impact of Binding Site Environment on the Optimization of TRPA1 Antagonists
11天前
已完结
Advances in TRP channel drug discovery: from target validation to clinical studies
14天前
已完结
Optimization of a Novel Quinazolinone-Based Series of Transient Receptor Potential A1 (TRPA1) Antagonists Demonstrating Potent in Vivo Activity
14天前
已完结
Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy
15天前
已完结
Discovery and SAR of JTE-151: A Novel RORγ Inhibitor for Clinical Development
17天前
已完结
Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease
18天前
已完结
Recent Advances in the Discovery of Oral TRPA1 Antagonists
23天前
已完结
Cationic Ester Prodrugs of Curcumin with N,N-dimethyl Amino Acid Promoieties Improved Poor Water Solubility and Intestinal Absorption
28天前
已完结
Synergistic Activity of Anticancer Polyphenols Embedded in Amphiphilic Dendrimer Nanoparticles
28天前
已完结
皖公网安备34019202002308
