Lv53
820 积分 2025-02-12 加入
Discovery of Potent and Selective Pyrrolo[2,3-d]pyrimidine Derivatives as Fourth-Generation EGFR Inhibitors Targeting Triple Mutations
33分钟前
已完结
Fragment-Based Discovery and Structure-Led Optimization of MSC778, the First Potent, Selective, and Orally Bioavailable FEN1 Inhibitor
2小时前
已完结
Discovery of Potent and Selective Reversible Ubiquitin-Like Modifier Activating Enzyme 5 Inhibitors Targeting the UFMylation Pathway
2小时前
已完结
Beyond Bioisosteres: Impact of Replacing a Benzene Ring with sp3-Rich Three-Dimensional Saturated Bridged Bicyclic Match Pairs on Biotransformation, Metabolic Stability, and Other ADME Profiles
2小时前
已完结
Direct Deaminative Halogenation at Hindered Tertiary Centers
4天前
已完结
Unlocking the power of affibody conjugated radioactive metallopharmaceuticals for targeted cancer diagnosis and therapy
4天前
已完结
Trithiol ligand provides tumor-targeting 191Pt-complexes with high molar activity and promising in vivo properties
22天前
已完结
A Highly Efficient Copper‐Mediated Radioiodination Approach Using Aryl Boronic Acids
1个月前
已完结
Discovery of Heteroaromatic Sulfones As a New Class of Biologically Compatible Thiol-Selective Reagents
2个月前
已完结
Tunable Heteroaromatic Sulfones Enhance in-Cell Cysteine Profiling
2个月前
已完结
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