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28 积分 2026-06-17 加入
Integrating Medicinal Chemist Expertise with Deep Learning for Automated Molecular Optimization
9小时前
已完结
Discovery of N-ethylpyridine-2-carboxamide derivatives as a novel scaffold for orally active γ-secretase modulators
1个月前
已完结
Optimization and biological evaluation of imidazopyridine derivatives as a novel scaffold for γ-secretase modulators with oral efficacy against cognitive deficits in Alzheimer’s disease model mice
1个月前
已完结
Exploring the chemical space of γ-secretase modulators
1个月前
已完结
Synthesis and Biological Activity of Flurbiprofen Analogues as Selective Inhibitors of β-Amyloid1-42Secretion
1个月前
已完结
Nonsteroidal anti-inflammatory drugs lower Aβ42 and change presenilin 1 conformation
1个月前
已完结
Selective inhibition of Aβ42 production by NSAID R‐enantiomers
1个月前
已完结
Applications of Bioisosteres in the Design of Biologically Active Compounds
2个月前
已完结