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26 积分 2025-02-11 加入
Identification of triazolyl KAT6 inhibitors via a templated fragment approach
18天前
已完结
Discovery of N-(2-oxoethyl) sulfanilamide-derived inhibitors of KAT6A (MOZ) against leukemia by an isostere strategy
20天前
已完结
Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents
21天前
已完结
Biological Activity and Structural Biology of Current KAT6A Inhibitor Chemotypes
22天前
已完结
Inhibitors of histone acetyltransferases KAT6A/B induce senescence and arrest tumour growth
22天前
已完结
Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A
22天前
已完结
Structure-based discovery of selective BRPF1 bromodomain inhibitors
23天前
已完结
RIMTAC: A Novel Degrader Design Platform by Indirect VHL-Recruitment via RIPK1
23天前
已完结
Discovery of Effective Dual PROTAC Degraders with Synergistic Antitumor Activity for Overcoming Tamoxifen-Resistant Breast Cancer
30天前
已完结
A Novel Dual-Targeting PROTAC Overcomes Endocrine Resistance by Engaging Orthosteric and Allosteric Sites of Estrogen Receptor α
30天前
已完结