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Late-Stage Lead Diversification Coupled with Quantitative Nuclear Magnetic Resonance Spectroscopy to Identify New Structure–Activity Relationship Vectors at Nanomole-Scale Synthesis: Application to Loratadine, a Human Histamine H1 Receptor Inverse Agonist
1小时前
求助中
Ppp2r1a Haploinsufficiency Increases Excitatory Synaptic Transmission and Decreases Spatial Learning by Impairing Endocannabinoid Signaling
4天前
已完结
Discovery of Novel P2Y 14 R Inhibitors for Ameliorating Liver Fibrosis by Suppressing Hepatic Stellate Cell Activation
6天前
已完结
Alicyclic Ring Size Variation of 4-Phenyl-2-naphthoic Acid Derivatives as P2Y14 Receptor Antagonists
6天前
已完结
Discovery of a Series of 4-Amide-thiophene-2-carboxyl Derivatives as Highly Potent P2Y14 Receptor Antagonists for Inflammatory Bowel Disease Treatment
6天前
已完结
Metabolism of the Antidepressant Mirtazapine in Vitro: Contribution of Cytochromes P-450 1A2, 2D6, and 3A4
19天前
已关闭
Mirtazapine revisited: new therapeutic perspectives and formulation advances
20天前
已完结
gem-Difluorobicyclo[2.1.1]hexanes via Photochemical [2π + 2σ] Cycloaddition Initiated by Oxidative Activation of gem-Difluorodienes
1个月前
已完结
Discovery of Novel, Potent, Selective, and Orally Available DGKα Inhibitors for the Treatment of Tumors
1个月前
已完结
Discovery of Fluoroalkenes as Dual Inhibitors of Diacylglycerol Kinases Alpha and Zeta (DGKα/ζ)
1个月前
已完结