Lv7
4920 积分 2023-10-02 加入
Ligand-embedded photoswitching PROTAC for spatiotemporal tubulin degradation
27天前
已完结
Discovery of novel pyridazinone derivatives as EGFRWT/ EGFRT790M kinase inhibitors; design, synthesis, antitumor evaluation, and molecular dynamic simulations
1个月前
已完结
Pharmaceutical applications of cyclopropyl containing scaffolds: a review on recent updates
1个月前
已完结
Design, synthesis, and antitumor evaluation of new pyridazinone scaffolds as dual EGFR/VEGFR-2 kinase inhibitors and apoptotic cells inducers
1个月前
已完结
Design, synthesis, and cytotoxicity screening of novel pyrazolopyrimidines over renal cell carcinoma (UO-31 cells) as p38α inhibitors, and apoptotic cells inducing activities
1个月前
已完结
Synthesis, characterization and antimicrobial activity of a series of substituted coumarin-3-carboxylatosilver(I) complexes
1个月前
已完结
Ligand-embedded photoswitching PROTAC for spatiotemporal tubulin degradation
2个月前
已完结
Novel imidazo[1,2-a]pyridine-based tubulin polymerization inhibitors: Structure-activity relationships and anti-tumor immune potentiation
2个月前
已完结
Discovery of the first dual PD-L1/JAK inhibitor with enhanced in vivo antitumor immunity
2个月前
已完结
Design, synthesis, and antiproliferative evaluation of dihydropyrimidinone-pyrazole derivatives as potential SHP2 inhibitors via in silico target prediction
3个月前
已完结