Lv3
210 积分 2024-08-08 加入
P2.10.17 Dual PARG-TOP1 Inhibition Exacerbates Dna-Protein Crosslinks and Replication Stress: A Promising Strategy for Enhancing Top1i-ADC Efficacy
4个月前
已关闭
Legumain-Cleavable Top1i Antibody-Drug Conjugates without Self-Immolative Spacers Demonstrate Potent Antitumor Activity
4个月前
已完结
Discovery and Preclinical Evaluation of PBX-7016, a Methylenedioxy-Camptothecin Payload for Antibody-Drug Conjugates with Enhanced Therapeutic Potential
4个月前
已完结
Neuraminidase-triggered activation of prodrug-type substrate of 4-nitroaniline
4个月前
已完结
Structure-Based Design and Synthesis of C-1- and C-4-Modified Analogs of Zanamivir as Neuraminidase Inhibitors
4个月前
已完结
A Practical Synthesis of Zanamivir Phosphonate Congeners with Potent Anti-influenza Activity
4个月前
已完结
Synthesis and anti-influenza activities of carboxyl alkoxyalkyl esters of 4-guanidino-Neu5Ac2en (zanamivir)
4个月前
已完结
Divalent oseltamivir analogues as potent influenza neuraminidase inhibitors
4个月前
已完结
Oseltamivir modified bovine serum albumin inhibits neuraminidase activity and accumulates virion particles to disturb influenza virus replication
4个月前
已完结
Cell surface clicking of antibody-recruiting polymers to metabolically azide-labeled cancer cells
5个月前
已完结