Lv7
3430 积分 2022-07-12 加入
Predictability of Idiosyncratic Drug Toxicity Risk for Carboxylic Acid-Containing Drugs Based on the Chemical Stability of Acyl Glucuronide
7天前
已完结
Early Process Development of a Heterobifunctional Protein Degrader
10天前
已完结
Rapid Identification of a Potent, Selective, and Orally Active p300/CBP Bromodomain Inhibitor Bearing an Imidazo[1,2- a ]pyridine Scaffold via a Highly Efficient Four-Step Synthesis
13天前
已完结
Discovery of BBI-355, a Potent, Selective, and Orally Available Checkpoint Kinase 1 Inhibitor for the Treatment of Extrachromosomal DNA Oncogene-Amplified Cancers
14天前
已关闭
Synthesis of 2-Aminophenols and Heterocycles by Ru-Catalyzed C–H Mono- and Dihydroxylation
16天前
已完结
Bicyclic Isosteres of Pyridine/Piperidine: From Synthesis to Applications
1个月前
已完结
Discovery of BT-114143, a Novel and Potent Phosphoric Acid-Containing Small-Molecule Plasminogen Activation Inhibitor for Hyperfibrinolysis
1个月前
已完结
An Efficient Synthesis of Ketone Enol Ethers Mediated byN-(1-Alkoxyalkyl)benzotriazoles
1个月前
已完结
Drug Delivery Strategy Exploiting Amino Acid Prodrugs: Improving Oral Bioavailability and Overcoming Nonlinear Pharmacokinetic Challenges Following Dose Escalation of a CK2 Inhibitor with Poor Solubility
1个月前
已完结
Chemical Ligand Space of Cereblon
1个月前
已完结