Lv4
716 积分 2025-09-22 加入
Conformationally Restricted Macrocycles as Improved FKBP51 Inhibitors Enabled by Systematic Linker Derivatization
16小时前
待确认
Conformationally Restricted Grp94-Selective Inhibitors
16小时前
待确认
Highly Conformationally Restricted Cyclopropane Tethers with Three-Dimensional Structural Diversity Drastically Enhance the Cell Permeability of Cyclic Peptides
16小时前
待确认
Influence of Hydrophobic Structures on the Plasma Membrane Permeability of Lipidlike Molecules
16小时前
待确认
Structure-Based Development of 3,4-Fused Tricyclic Benzofuran Derivatives as Polyketide Synthase 13 Inhibitors with Negligible hERG Inhibition
16小时前
待确认
Late-stage functionalization with strain-release warheads enables tunable covalent inhibition
21天前
已完结
Characterising covalent warhead reactivity
25天前
已完结
Application of Bioisosteres in the Design and Discovery of FDA-Approved Drugs and Advanced Clinical Candidates
1个月前
已完结
Synthesis and Pharmacological Activities of Pyrazole Derivatives: A Review
3个月前
已完结
An Overview of the Pharmacological Activities and Synthesis of Benzothiophene Derivatives
3个月前
已完结