Lv11
100 积分 2025-09-05 加入
Design, synthesis and biological activity evaluation of novel allosteric inhibitors of the DENV NS2B–NS3 protease
8个月前
已完结
Discovery of Highly Potent, Selective, and Orally Efficacious p300/CBP Histone Acetyltransferases Inhibitors
9个月前
已完结
Early Drug‐Discovery Efforts towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors
9个月前
已完结
Discovery, Structure–Activity Relationship, and Biological Activity of Histone-Competitive Inhibitors of Histone Acetyltransferases P300/CBP
9个月前
已完结
Discovery of NVP-BYL719 a potent and selective phosphatidylinositol-3 kinase alpha inhibitor selected for clinical evaluation
9个月前
已完结
Histone acetyltransferase inhibitors: An overview in synthesis, structure-activity relationship and molecular mechanism
10个月前
已完结
Molecular Docking and Simulation Studies Predict Lactyl-CoA as the Substrate for P300 Directed Lactylation
10个月前
已完结
Discovery of DS-9300: A Highly Potent, Selective, and Once-Daily Oral EP300/CBP Histone Acetyltransferase Inhibitor
10个月前
已完结
Discovery of CPI-1612: A Potent, Selective, and Orally Bioavailable EP300/CBP Histone Acetyltransferase Inhibitor
10个月前
已完结
The structural basis of protein acetylation by the p300/CBP transcriptional coactivator
10个月前
已完结