Lv6
2840 积分 2024-03-04 加入
Carbonylative Ring Expansion of Cyclic Carboxylic Acids
26天前
已完结
Synthesis and Structure-Activity Relationships of Novel Retinoid X Receptor-Selective Retinoids
1个月前
已完结
4-[3-(4-Cyclopropanecarbonylpiperazine-1-carbonyl)-4-fluorobenzyl]-2H-phthalazin-1-one: A Novel Bioavailable Inhibitor of Poly(ADP-ribose) Polymerase-1
1个月前
已完结
Discovery of 4-Amino-N-[(1S)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide (AZD5363), an Orally Bioavailable, Potent Inhibitor of Akt Kinases
1个月前
已完结
Electrophilic Cyanation of Boron Enolates: Efficient Access to Various β‐Ketonitrile Derivatives
1个月前
已完结
Journey of Methionine Adenosyltransferase 2A Inhibitors: From Bench to Advanced Clinical Trials
3个月前
已完结
Discovery of AG-270, a First-in-Class Oral MAT2A Inhibitor for the Treatment of Tumors with Homozygous MTAP Deletion
3个月前
已完结
Covalent inhibitors of human cytochrome P450 3A4: research advances and future perspectives
3个月前
已完结
Development of a Generalized, Quantitative Physicochemical Model of CYP3A4 Inhibition for Use in Early Drug Discovery
3个月前
已完结
Linker Design for Antibody–Drug Conjugates
4个月前
已完结