Lv7
3370 积分 2024-03-04 加入
Insights into interferon regulatory factor activation from the crystal structure of dimeric IRF5
13天前
已完结
Covalent Degraders of Immune Regulatory Transcription Factors IRF8 and IRF5
27天前
已完结
SH-1028, An Irreversible Third-Generation EGFR TKI, Overcomes T790M-Mediated Resistance in Non-Small Cell Lung Cancer
28天前
已完结
Biological Activity and Structural Biology of Current KAT6A Inhibitor Chemotypes
2个月前
已完结
Carbonylative Ring Expansion of Cyclic Carboxylic Acids
3个月前
已完结
Synthesis and Structure-Activity Relationships of Novel Retinoid X Receptor-Selective Retinoids
4个月前
已完结
4-[3-(4-Cyclopropanecarbonylpiperazine-1-carbonyl)-4-fluorobenzyl]-2H-phthalazin-1-one: A Novel Bioavailable Inhibitor of Poly(ADP-ribose) Polymerase-1
4个月前
已完结
Discovery of 4-Amino-N-[(1S)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide (AZD5363), an Orally Bioavailable, Potent Inhibitor of Akt Kinases
4个月前
已完结
Electrophilic Cyanation of Boron Enolates: Efficient Access to Various β‐Ketonitrile Derivatives
4个月前
已完结
Journey of Methionine Adenosyltransferase 2A Inhibitors: From Bench to Advanced Clinical Trials
5个月前
已完结