Lv681
2720 积分 2023-03-01 加入
Structure-Guided Conformational Restriction Leading to High-Affinity, Selective, and Cell-Active Tetrahydroisoquinoline-Based Noncovalent Keap1-Nrf2 Inhibitors
1个月前
已完结
Discovery of Casdatifan, Part I: Design and Characterization of Tetrahydroquinoline Inhibitors of Hypoxia-Inducible Factor-2α
2个月前
已完结
Identification of gp120 Residue His105 as a Novel Target for HIV-1 Neutralization by Small-Molecule CD4-Mimics
2个月前
已完结
Visible Light Mediated Chemoselective Hydroxylation of Benzylic Methylenes
2个月前
已完结
Deoxygenative Asymmetric Cyanation with P(OEt)3 Employing Cooperative Photoredox Catalysis and Copper Catalysis
4个月前
已完结
Single-Dose Oral Influenza Antiviral Prodrug Enabled by Cholesterol Conjugation
9个月前
已完结
Triazoles in Medicinal Chemistry: Physicochemical Properties, Bioisosterism, and Application
10个月前
已完结
Medoxomil Prodrug Strategies
1年前
已完结