Lv42
545 积分 2021-01-05 加入
Discovery of Kinesin KIF18A Inhibitor ATX020: Tactical Application of Silicon Atom Replacement
12小时前
已完结
Syntheses of Potent, Selective, and Orally Bioavailable Indazole-Pyridine Series of Protein Kinase B/Akt Inhibitors with Reduced Hypotension
1天前
已完结
Beyond Inhibition: Recent Advances of Heterobifunctional Molecules Targeting CDK9
1天前
已完结
Macrocyclic-based strategy in drug design: From lab to the clinic
5天前
已完结
The Ugi Multicomponent Reaction for the One‐Step Construction of Macrocycles
5天前
已完结
2-Aminothiadiazole inhibitors of AKT1 as potential cancer therapeutics
5天前
已完结
Optimization of microtubule affinity regulating kinase (MARK) inhibitors with improved physical properties
6天前
已完结
Discovery of Dual CDK6/PIM1 Inhibitors with a Novel Structure, High Potency, and Favorable Druggability for the Treatment of Acute Myeloid Leukemia
6天前
已完结
Discovery of Peptide Boronate Derivatives as Histone Deacetylase and Proteasome Dual Inhibitors for Overcoming Bortezomib Resistance of Multiple Myeloma
6天前
已完结
Structure-Based Macrocycle Design in Small-Molecule Drug Discovery and Simple Metrics To Identify Opportunities for Macrocyclization of Small-Molecule Ligands
6天前
已完结