Lv11
2 积分 2022-08-29 加入
TAS‐120 Cancer Target Binding: Defining Reactivity and Revealing the First Fibroblast Growth Factor Receptor 1 (FGFR1) Irreversible Structure
1小时前
已完结
Discovery of Reversible Covalent Bruton’s Tyrosine Kinase Inhibitors PRN473 and PRN1008 (Rilzabrutinib)
1小时前
已完结
Discovery of Affinity‐Based Probes for Btk Occupancy Assays
1小时前
已完结
Design, Structure Optimization, and Preclinical Characterization of JAB-21822, a Covalent Inhibitor of KRASG12C
1小时前
已完结
Quantitative Evaluation of Each Catalytic Subsite of Cathepsin B for Inhibitory Activity Based on Inhibitory Activity–Binding Mode Relationship of Epoxysuccinyl Inhibitors by X-ray Crystal Structure Analyses of Complexes
1小时前
已完结
Revealing the limits of covalent docking and advancing affinity prediction with covalent-aware multi-task learning
21天前
已完结
CovalentInDB: a comprehensive database facilitating the discovery of covalent inhibitors
1个月前
已完结
A practical guide to large-scale docking
1个月前
已完结
Chemical Space Exploration of a Database of Covalent Binders in the PDB
1个月前
已关闭
Transition Metal Nanoparticle Catalysis in Ionic Liquids
6个月前
已完结