铑
化学
芳基
催化作用
苯并噻嗪
三环
药物化学
组合化学
立体化学
有机化学
烷基
作者
Gao Huang,Yujia Shan,Jin‐Tao Yu,Changduo Pan
摘要
The synthesis of 1,2-benzothiazine derivatives through rhodium-catalyzed C-H activation/cyclization of S-aryl sulfoximines with iodonium ylides was developed for the first time. In this report, C-H and N-H bond functionalization was realized towards a series of tricyclic and tetracyclic sulfoximine derivatives with moderate to excellent yields under simple reaction conditions.
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