化学
烷基化
有机化学
胺化
脱碳
药物化学
反应条件
组合化学
炔烃
还原胺化
作者
Kelu Yan,Xiaoyu Wang,Jiangwei Wen,Jianjing Yang,Yuanyuan Zhang,Bingxin Zhou,Daoshan Yang
摘要
A chelate-assisted copper-catalyzed 1,2-alkylamidation of alkynes with aldehydes and amides have been proposed. The generation of high-capacity alkylated enamides exhibits stubborn anti -stereoselectivity and β-regioselectivity.
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