Synthesis of 2-glycosyl-quinazolines and 5-glycosyl-pyrazolo[1,2-a]cinnolines by Cp*Ir(III)-catalyzed C-H activation/cyclization

A novel strategy for the synthesis of 2-glycosyl-quinazolines and 5-glycosyl-pyrazolo[1,2-a]cinnolines has been established through an Ir-catalyzed C-H activation/annulation process. This approach features mild reaction conditions, exhibits good tolerance to diverse...