Structure-guided discovery of a novel, potent, and orally bioavailable 3,5-dimethylisoxazole aryl-benzimidazole BET bromodomain inhibitor
作者
David Sperandio,Vangelis Aktoudianakis,Kerim Babaoglu,Xiaowu Chen,Kristyna M. Elbel,Gregory Chin,Britton K. Corkey,Jinfa Du,Bob Jiang,Tetsuya Kobayashi,Richard L. Mackman,Ruben Martinez,Hai Yang,Jeff Zablocki,Saritha Kusam,Kim Jordan,Heather K. Webb,Jamie Bates,Latesh Lad,Michael Mish