化学
共域化
细胞生物学
生物素化
荧光
受体
烟碱乙酰胆碱受体
生物化学
炎症
乙酰胆碱受体
生物物理学
荧光团
抑制性突触后电位
分子生物学
细胞内
炎症性肠病
寡肽
肽
分子探针
淀粉样蛋白(真菌学)
共核细胞病
作用机理
紧身衣
作者
Yao Tan,Tao Ma,Songze Li,Chenxing Xu,Yu Han,dongting zhangsun,Xuetao Zhu,Sulan Luo
标识
DOI:10.1021/acs.jmedchem.5c03269
摘要
The α7 nicotinic acetylcholine receptor (α7 nAChR) modulates neuroimmune signaling but remains poorly characterized in peripheral disease due to a lack of visualization tools. We developed the fluorescent probe LvID-BDP by conjugating a BODIPY fluorophore to the high-affinity α7 nAChR-targeting peptide LvID. LvID-BDP showed high quantum yield, robust photostability, and sufficient physiological stability for biological imaging. Electrophysiology characterized LvID-BDP as a potent α7 nAChR antagonist, exhibiting a half-maximal inhibitory concentration (IC50) of 119.2 nM while retaining high affinity and specificity for the receptor. In murine colon sections, LvID-BDP specifically labeled α7 nAChR, showing strong antibody colocalization (Pearson's R = 0.87) while revealing macrophage-selective enrichment (Pearson's R = 0.85). This probe detected α7 nAChR alterations in engineered and inflamed macrophages and quantified its expression in inflammatory bowel disease (IBD) tissues. LvID-BDP provides a valuable pharmacological tool for specific α7 nAChR visualization in peripheral disease contexts, advancing pathological mechanism research.
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