细胞内
化学
环肽
小分子
计算生物学
组合化学
药物发现
肽
纳米技术
生物化学
生物
材料科学
作者
Atsushi Ohta,Mikimasa Tanada,Shojiro Shinohara,Yuya Morita,Kazuhiko Nakano,Y. Yamagishi,Ryusuke Takano,Shiori Kariyuki,Takeo Iida,Atsushi Matsuo,Kazuhisa Ozeki,Takashi EMURA,Yuuji Sakurai,Koji Takano,Atsuko Higashida,Miki Kojima,Terushige Muraoka,Ryuuichi Takeyama,Tatsuya Kato,Kaori Kimura
摘要
-alkylated cyclic peptide hits. We discovered a KRAS inhibitory clinical compound (LUNA18) as the first example of our platform technology.
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