Metal-Free Stereoselective C(sp3)-H Indolation of N-heterocycles to Potent Antimicrobial Non-Canonical Tryp-Pro Hybrids

Indolyl aliphatic N-heterocycles are widely present as the key structural unit of many natural products and unnatural bioactive molecules. The known synthetic methods of indolyl N-heterocycles rely on metallic reagents/catalysts,...