Rapid hit to lead evaluation of pyrazolo[3,4-d]pyrimidin-4-one as selective and orally bioavailable mGluR1 antagonists
作者
Xueqing Wang,Teodozyi Kolasa,Odile F. El Kouhen,Linda E. Chovan,Candace L. Black-Shaefer,Frank L. Wagenaar,Jennifer A. Garton,Robert B. Moreland,Prisca Honoré,Yau Yi Lau,Peter J. Dandliker,Jorge D. Brioni,Andrew O. Stewart