医学
埃罗替尼
内科学
药理学
肿瘤科
毒性
胃肠病学
作者
Akinobu Hamada,Yuki Kai,Jiichiro Sasaki,Sho Saeki,Hiroto Kishi,Shinji Fujii,Hiroshi Semba,Takeshi Isobe,Yutaka Hashimoto,Hirotsugu Kohrogi,Hideyuki Saito
标识
DOI:10.1200/jco.2012.30.15_suppl.e13072
摘要
e13072 Background: Erlotinib is metabolized by cytochrome P450 enzymes to form a para-hydroxyaniline metabolite that is further metabolized to quinone-imine. Erlotinib is detoxified when it conjuga...
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