| 标题 |
Discovery of 2-(6-{[(1R,2R)-2-hydroxycyclohexyl]amino}-4,5-dimethylpyridazin-3-yl)-5-(trifluoromethyl)phenol (ASP0965): A potent, orally active and brain-penetrable NLRP3 inflammasome inhibitor with a novel scaffold for the treatment of α-synucleinopathy |
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| DOI | |
| 其它 |
期刊:Bioorganic & Medicinal Chemistry 作者:Yusuke Inagaki; Takashi Kamikubo; Ikumi Kuriwaki; Junko Watanabe; Susumu Yamaki; et al 出版日期:2024-12-12 |
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(2025-6-4)