炎症体
脂多糖
目标2
半胱氨酸蛋白酶1
败血症
药理学
基因敲除
化学
过氧化物还原蛋白
姜黄素
医学
炎症
生物化学
免疫学
细胞凋亡
酶
过氧化物酶
作者
Wen Liu,Wenjie Guo,Yongcheng Zhu,Shuang Peng,Wei Zheng,Chao Zhang,Fenli Shao,Yuyu Zhu,Nan Hang,Ling‐Dong Kong,Xiangbao Meng,Qiang Xu,Yang Sun
出处
期刊:Journal of Immunology
[American Association of Immunologists]
日期:2018-09-05
卷期号:201 (8): 2403-2413
被引量:45
标识
DOI:10.4049/jimmunol.1700796
摘要
Aberrant activation of the NLRP3 inflammasome contributes to the onset and progression of various inflammatory diseases, making it a highly desirable drug target. In this study, we screened a series of small compounds with anti-inflammatory activities and identified a novel NLRP3 inflammasome inhibitor, AI-44, a curcumin analogue that selectively inhibited signal 2 but not signal 1 of NLRP3 inflammasome activation. We demonstrated that AI-44 bound to peroxiredoxin 1 (PRDX1) and promoted the interaction of PRDX1 with pro-Caspase-1 (CASP1), which led to the suppression of association of pro-CASP1 and ASC. Consequently, the assembly of the NLRP3 inflammasome was interrupted, and the activation of CASP1 was inhibited. Knockdown of PRDX1 significantly abrogated the inhibitory effect of AI-44 on the NLRP3 inflammasome. Importantly, AI-44 alleviated LPS-induced endotoxemia in mice via suppressing NLRP3 inflammasome activation. Taken together, our work highlighted PRDX1 as a negative regulator of NLRP3 inflammasome activation and suggested AI-44 as a promising candidate compound for the treatment of sepsis or other NLRP3 inflammasome-driven diseases.
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